SCHEMBL6578728

SCHEMBL6578728

COc1cc(C(=O)NN)ccc1OCc1ccccc1

nearest known ligand 0.76

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.73
ALDH1A1 P00352 1/20 0.73
MAPT P10636 1/20 0.73
SMPD1 P17405 3/20 0.72
HDAC1 Q13547 1/20 0.72
HDAC8 Q9BY41 1/20 0.72
HDAC6 Q9UBN7 1/20 0.72
MEN1 O00255 1/20 0.70
KMT2A Q03164 1/20 0.70
NPC1 O15118 4/20 0.70
RAB9A P51151 4/20 0.70
HPGD P15428 1/20 0.70
SMN1; SMN2 Q16637 1/20 0.70
MRGPRX4 Q96LA9 1/20 0.59
RXRA P19793 1/20 0.58
CASP3 P42574 1/20 0.57
SENP7 Q9BQF6 1/20 0.57
ATM Q13315 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584177 0.95 SMPD1 (0.81) KDM4EALDH1A1MAPTSMPD1HDAC1
SCHEMBL24077087 0.89 SMPD1 (0.72) KDM4EALDH1A1MAPTSMPD1HDAC1
SCHEMBL28325672 0.89 SMPD1 (0.90) KDM4ESMPD1HDAC1HDAC8HDAC6
SCHEMBL4278415 0.86 NPC1 (0.73) KDM4EALDH1A1MAPTSMPD1HDAC1
SCHEMBL2063068 0.86 SMN1; SMN2 (0.73) KDM4EALDH1A1MAPTSMPD1HDAC1
SCHEMBL242563 0.86 MRGPRX4 (0.77) KDM4ESMPD1HDAC1HDAC8HDAC6
SCHEMBL27881765 0.86 NPC1 (0.77) KDM4EMAPTSMPD1HDAC1HDAC8
SCHEMBL7237622 0.85 ALDH1A1 (0.63) KDM4EALDH1A1MAPTSMPD1HDAC1
SCHEMBL11277266 0.85 MRGPRX4 (0.75) KDM4ESMPD1HDAC1HDAC8HDAC6
SCHEMBL31025721 0.85 NPC1 (0.75) KDM4EMAPTSMPD1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1148357-C Triazole and imidazole derivative - 2004-05-05 CN disclosed
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
CN-1281852-A Triazole and imidazole derivative HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed