SCHEMBL6579157

SCHEMBL6579157

Nc1ccccc1-c1c(N)c(-c2ccccc2N)c(-c2ccccc2N)c(N)c1-c1ccccc1N

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.67
L3MBTL1 Q9Y468 3/20 0.67
HSD17B10 Q99714 1/20 0.55
ALOX15 P16050 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
CYP3A4 P08684 1/20 0.50
CASP1 P29466 1/20 0.50
CASP7 P55210 1/20 0.50
ADORA2A P29274 3/20 0.44
PTPRC P08575 1/20 0.44
MAOA P21397 2/20 0.44
FGR P09769 1/20 0.44
PIM1 P11309 1/20 0.44
CSNK1A1 P48729 1/20 0.44
CSNK1D P48730 1/20 0.44
DYRK1A Q13627 1/20 0.44
HIPK2 Q9H2X6 1/20 0.44
CSNK1G1 Q9HCP0 1/20 0.44
MAOB P27338 1/20 0.41
IDO1 P14902 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5146944 0.92 ALDH1A1 (0.63) ALDH1A1L3MBTL1HSD17B10ALOX15SMN1; SMN2
SCHEMBL3174480 0.86 ALDH1A1 (0.60) ALDH1A1L3MBTL1HSD17B10ALOX15SMN1; SMN2
SCHEMBL5517538 0.86 ALDH1A1 (0.63) ALDH1A1L3MBTL1HSD17B10ALOX15SMN1; SMN2
SCHEMBL7389021 0.82 ALDH1A1 (0.67) ALDH1A1L3MBTL1HSD17B10ALOX15SMN1; SMN2
SCHEMBL169281 0.81 ALDH1A1 (1.00) ALDH1A1L3MBTL1HSD17B10ALOX15SMN1; SMN2
SCHEMBL31607672 0.81 ALDH1A1 (1.00) ALDH1A1L3MBTL1HSD17B10ALOX15SMN1; SMN2
SCHEMBL3714036 0.80 ALDH1A1 (0.72) ALDH1A1L3MBTL1HSD17B10ALOX15SMN1; SMN2
SCHEMBL4798865 0.80 ALDH1A1 (0.63) ALDH1A1L3MBTL1HSD17B10ALOX15SMN1; SMN2
SCHEMBL5493737 0.78 ALDH1A1 (0.68) ALDH1A1L3MBTL1HSD17B10ALOX15SMN1; SMN2
Ammonia Solution, Strong SCHEMBL21297045 0.78 ALDH1A1 (0.93) ALDH1A1L3MBTL1HSD17B10ALOX15SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090910-B1 AMINIUM SALT OR DIIMONIUM SALT COMPOUNDS AND USE THEREOF NIPPON KAYAKU KK (JP) 2004-09-29 EP claimed
EP-1090910-A1 AMMINIUM SALT OR DIIMMONIUM SALT COMPOUNDS AND USE THEREOF Nippon Kayaku Kabushiki Kaisha (JP) 2001-04-11 EP claimed
EP-1090910-B1 AMINIUM SALT OR DIIMONIUM SALT COMPOUNDS AND USE THEREOF NIPPON KAYAKU KK (JP) 2004-09-29 EP disclosed
US-6475590-B1 OPTICAL RECORDING MEDIUM OR THE INFRARED RAY SCREENING FILTER. NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2002-11-05 US disclosed
EP-1090910-A1 AMMINIUM SALT OR DIIMMONIUM SALT COMPOUNDS AND USE THEREOF Nippon Kayaku Kabushiki Kaisha (JP) 2001-04-11 EP disclosed