SCHEMBL6579386

SCHEMBL6579386

COc1ccc(C2=NN(C(=O)c3cccc(NC(=O)c4ccc(N)cc4)c3)CCC2)cc1OC(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
NPSR1 Q6W5P4 2/20 0.43
LMNA P02545 2/20 0.43
PKM P14618 1/20 0.43
POLB P06746 1/20 0.43
PGR P06401 8/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
MAOB P27338 1/20 0.41
KDM4E B2RXH2 1/20 0.39
ATM Q13315 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
MEN1 O00255 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581799 0.90 NPC1 (0.45) ALDH1A1NPSR1LMNAPKMPOLB
SCHEMBL6584543 0.88 PDE5A (0.52) MEN1MAPK1KMT2A
SCHEMBL3921987 0.88 ALDH1A1 (0.52) ALDH1A1NPSR1LMNAPKMPOLB
SCHEMBL6583317 0.88 PGR (0.49) ALDH1A1LMNAPGRNPC1RAB9A
SCHEMBL5206295 0.87 ALDH1A1 (0.49) ALDH1A1NPSR1LMNAPKMPOLB
SCHEMBL6602100 0.85 MAOB (0.48) ALDH1A1NPSR1LMNAPKMPOLB
Hydrochloric Acid SCHEMBL7646213 0.84 MAOB (0.47) ALDH1A1NPSR1LMNAPKMPOLB
SCHEMBL6583658 0.83 NPC1 (0.45) ALDH1A1NPSR1LMNAPKMPOLB
SCHEMBL6581923 0.82 NPC1 (0.48) ALDH1A1NPSR1LMNAPKMPOLB
SCHEMBL6582371 0.82 NPC1 (0.49) ALDH1A1NPSR1LMNAPKMPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194411-B1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2004-06-16 EP disclosed
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed