SCHEMBL6579659

SCHEMBL6579659

CC(C)(C)OC(=O)N1CCN(CCCC(Oc2cc(Cl)ccc2Cl)c2ccccc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 3/20 0.49
CNR1 P21554 1/20 0.42
OPRM1 P35372 1/20 0.42
OPRL1 P41146 1/20 0.42
ACKR3 P25106 3/20 0.42
CYP3A4 P08684 1/20 0.42
CYP3A5 P20815 1/20 0.42
HTR1A P08908 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ABCB1 P08183 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6502752 0.84 NOS2 (0.58) NOS2CYP3A4CYP3A5HTR1A
SCHEMBL6576553 0.79 NOS2 (0.53) NOS2OPRM1OPRL1
SCHEMBL6576611 0.78 NOS2 (0.55) NOS2OPRM1OPRL1
Fumaric Acid SCHEMBL6579320 0.78 NOS2 (0.61) NOS2OPRM1OPRL1MEN1KMT2A
Fumaric Acid SCHEMBL6579315 0.78 NOS2 (0.61) NOS2OPRM1OPRL1MEN1KMT2A
Fumaric Acid SCHEMBL6577450 0.77 NOS2 (0.60) NOS2OPRM1OPRL1MEN1KMT2A
Fumaric Acid SCHEMBL6577457 0.77 NOS2 (0.60) NOS2OPRM1OPRL1MEN1KMT2A
SCHEMBL6577453 0.76 NOS2 (0.52) NOS2OPRM1OPRL1CYP3A4MEN1
SCHEMBL31420190 0.74 SLC6A4 (0.62) OPRM1CYP3A4HTR1AMEN1KMT2A
SCHEMBL15567036 0.73 KMT2A (0.50) CNR1ACKR3CYP3A4CYP3A5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6743939-B2 NITRIC OXIDE SYNTHASE INHIBITORS; SUCH AS 4-CHLORO-2-(((1)-4-(METHYLAMINO)-1-PHENYLBUTYL)OXY)BENZONITRILE ASTRAZENECA AB (SE) 2004-06-01 US disclosed
EP-1263714-B1 NOVEL PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2004-04-28 EP disclosed
US-20030105161-A1 Novel phenylheteroalkylamine derivatives ASTRAZENECA AB (SE) 2003-06-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030105161-A1 Novel phenylheteroalkylamine derivatives NOS1, CYP1A1, NOS2 NOS2 3/4885CNR1 144/4885OPRM1 8/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.