SCHEMBL6580820

SCHEMBL6580820

COC(=O)c1ccc(CN2CCCC2)s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.49
ALDH1A1 P00352 3/20 0.48
HPGD P15428 2/20 0.48
KDM4E B2RXH2 2/20 0.47
NPSR1 Q6W5P4 3/20 0.47
L3MBTL1 Q9Y468 3/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PARP1 P09874 1/20 0.46
LMNA P02545 1/20 0.45
PPARG P37231 1/20 0.45
NCOA2 Q15596 1/20 0.45
NCOA1 Q15788 1/20 0.45
NCOA3 Q9Y6Q9 1/20 0.45
MRGPRX4 Q96LA9 1/20 0.45
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
ATM Q13315 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3823243 0.88 HRH3 (0.60) HRH3SMN1; SMN2ALDH1A1HPGDKDM4E
SCHEMBL16761062 0.87 ALDH1A1 (0.54) HRH3ALDH1A1HPGDNPSR1L3MBTL1
SCHEMBL8177110 0.85 HRH3 (0.55) HRH3SMN1; SMN2ALDH1A1HPGDKDM4E
SCHEMBL3592586 0.85 HRH3 (0.57) HRH3ALDH1A1HPGDKDM4EL3MBTL1
SCHEMBL8184741 0.83 HRH3 (0.61) HRH3SMN1; SMN2ALDH1A1HPGDKDM4E
Hydrochloric Acid SCHEMBL8176778 0.83 HRH3 (0.58) HRH3SMN1; SMN2ALDH1A1HPGDKDM4E
SCHEMBL6578561 0.81 HRH3 (0.53) HRH3ALDH1A1HPGDKDM4EL3MBTL1
SCHEMBL8171401 0.80 HRH3 (0.55) HRH3SMN1; SMN2ALDH1A1HPGDKDM4E
SCHEMBL8179534 0.79 HRH3 (0.58) HRH3SMN1; SMN2ALDH1A1HPGDKDM4E
SCHEMBL8178308 0.79 HRH3 (0.58) HRH3SMN1; SMN2ALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed