SCHEMBL6580942

SCHEMBL6580942

COc1ccc(-c2nc(-c3cccc(CN(C)C)c3)n[nH]2)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.46
ADORA2A P29274 3/20 0.46
ADORA1 P30542 2/20 0.46
NR1H2 P55055 1/20 0.46
NR1H3 Q13133 1/20 0.46
LCK P06239 2/20 0.44
BTK Q06187 2/20 0.44
S1PR1 P21453 2/20 0.44
TLR8 Q9NR97 2/20 0.43
TLR7 Q9NYK1 2/20 0.43
TLR9 Q9NR96 1/20 0.43
KDM4E B2RXH2 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CSF1R P07333 1/20 0.42
ACHE P22303 1/20 0.40
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6581027 0.99 HTR7 (0.46) HTR7ADORA2AADORA1NR1H2NR1H3
SCHEMBL6578288 0.90 S1PR1 (0.47) HTR7ADORA2AADORA1NR1H2NR1H3
Hydrochloric Acid SCHEMBL6581197 0.89 S1PR1 (0.53) HTR7ADORA2AADORA1NR1H2NR1H3
Hydrochloric Acid SCHEMBL6578720 0.89 S1PR1 (0.46) HTR7ADORA2AADORA1NR1H2NR1H3
SCHEMBL6581627 0.89 S1PR1 (0.42) HTR7ADORA2AADORA1NR1H2NR1H3
Hydrochloric Acid SCHEMBL6581348 0.88 S1PR1 (0.41) HTR7ADORA2AADORA1NR1H2NR1H3
SCHEMBL6578750 0.87 NR1H2 (0.47) HTR7ADORA2AADORA1NR1H2NR1H3
Hydrochloric Acid SCHEMBL6578160 0.86 NR1H2 (0.46) HTR7ADORA2AADORA1NR1H2NR1H3
Hydrochloric Acid SCHEMBL6580524 0.82 NR1H2 (0.58) HTR7ADORA2AADORA1NR1H2NR1H3
SCHEMBL6578503 0.82 ADORA2A (0.62) HTR7ADORA2AADORA1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP claimed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US claimed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP claimed
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed