SCHEMBL6580950

SCHEMBL6580950

CCOc1cc(C2=NN(C(=O)c3cccc(NC(=O)c4ccc(NC(=O)c5cccc(OC)c5)cc4)c3)CCC2)ccc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.45
RAB9A P51151 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
KMT2A Q03164 6/20 0.45
MEN1 O00255 4/20 0.45
MAPT P10636 3/20 0.45
ALDH1A1 P00352 3/20 0.45
POLB P06746 2/20 0.45
LMNA P02545 2/20 0.45
QSOX1 O00391 1/20 0.45
PKM P14618 1/20 0.45
KDM4E B2RXH2 1/20 0.45
USP2 O75604 1/20 0.45
NR1H4 Q96RI1 1/20 0.44
IDO1 P14902 1/20 0.43
TDO2 P48775 1/20 0.43
TP53 P04637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6767556 0.98 ALDH1A1 (0.47) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL7557662 0.96 NPC1 (0.44) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6585136 0.96 ALDH1A1 (0.49) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6763155 0.95 ALDH1A1 (0.51) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6583333 0.95 KMT2A (0.49) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6585175 0.95 ALDH1A1 (0.51) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6584808 0.94 NPC1 (0.50) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6581923 0.94 NPC1 (0.48) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6581435 0.93 KMT2A (0.49) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6583265 0.93 NPC1 (0.45) NPC1RAB9ASMN1; SMN2NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194411-B1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2004-06-16 EP disclosed
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed