SCHEMBL6763155

SCHEMBL6763155

CCOc1cc(C2=NN(C(=O)c3ccc(NC(=O)c4cccc(NC(=O)c5ccc(OC)cc5)c4)cc3)CCC2)ccc1OC

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
POLB P06746 2/20 0.51
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 1/20 0.47
NPC1 O15118 6/20 0.47
KMT2A Q03164 6/20 0.47
MEN1 O00255 5/20 0.47
RAB9A P51151 4/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
TP53 P04637 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPT P10636 2/20 0.44
PLAU P00749 1/20 0.43
LMNA P02545 1/20 0.43
GAA P10253 1/20 0.42
CASP1 P29466 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6585175 0.97 ALDH1A1 (0.51) ALDH1A1POLBCYP1A2CYP3A4NPC1
SCHEMBL6767556 0.95 ALDH1A1 (0.47) ALDH1A1POLBCYP1A2CYP3A4NPC1
SCHEMBL6581435 0.95 KMT2A (0.49) ALDH1A1POLBNPC1KMT2AMEN1
SCHEMBL6580950 0.95 NPC1 (0.45) ALDH1A1POLBCYP1A2CYP3A4NPC1
SCHEMBL6584808 0.95 NPC1 (0.50) ALDH1A1POLBCYP1A2NPC1KMT2A
SCHEMBL6581784 0.94 ALDH1A1 (0.55) ALDH1A1POLBCYP1A2NPC1KMT2A
SCHEMBL6584628 0.94 PGR (0.47) ALDH1A1POLBNPC1KMT2AMEN1
SCHEMBL6585136 0.94 ALDH1A1 (0.49) ALDH1A1POLBNPC1KMT2AMEN1
SCHEMBL6583333 0.94 KMT2A (0.49) ALDH1A1POLBNPC1KMT2AMEN1
SCHEMBL6581858 0.93 SMN1; SMN2 (0.49) ALDH1A1POLBCYP1A2NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed