SCHEMBL658101

SCHEMBL658101

CC(=O)c1c(O)cc(OCc2ccccc2)cc1OCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.61
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.51
CYP2C19 P33261 2/20 0.51
MAPT P10636 1/20 0.51
CYP2C9 P11712 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
CASP3 P42574 1/20 0.51
SENP8 Q96LD8 1/20 0.51
SENP7 Q9BQF6 1/20 0.51
SENP6 Q9GZR1 1/20 0.51
USP2 O75604 1/20 0.50
CYP3A4 P08684 1/20 0.50
MAPK1 P28482 1/20 0.50
CA9 Q16790 1/20 0.50
SLC5A1 P13866 1/20 0.49
SLC5A2 P31639 1/20 0.49
BRD4 O60885 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30141054 1.00 MAOB (0.61) MAOBMEN1KMT2ASMN1; SMN2CYP2C19
SCHEMBL11739144 0.92 MAOB (0.59) MAOBMEN1KMT2ASMN1; SMN2CYP2C19
SCHEMBL14178903 0.92 CYP3A4 (0.63) MAOBMEN1KMT2ASMN1; SMN2MAPT
SCHEMBL14181066 0.91 MAOB (0.68) MAOBMEN1KMT2ASMN1; SMN2CYP2C19
SCHEMBL18526952 0.91 MAOB (0.51) MAOBMEN1KMT2ASMN1; SMN2CYP2C19
SCHEMBL14616693 0.90 MAOB (0.56) MAOBMEN1KMT2ASMN1; SMN2CYP2C19
SCHEMBL30789227 0.90 MAOB (0.56) MAOBMEN1KMT2ASMN1; SMN2CYP2C19
SCHEMBL14178921 0.87 MAOB (0.54) MAOBMEN1KMT2ASMN1; SMN2L3MBTL1
SCHEMBL26455213 0.87 MAOB (0.54) MAOBMEN1KMT2ASMN1; SMN2CYP2C19
SCHEMBL10147478 0.87 MAPT (0.53) MAOBSMN1; SMN2CYP2C19MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 72 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100048920-A1 Preparation of (+)-Catechin, (-)-Epicatechin, (-)-Catechin, and (+)-Epicatechin and Their 5,7,3',4'-Tetra-O-Benzyl Analogues MARS, INCORPORATED (US) 2010-02-25 US claimed
EP-1896443-A1 PREPARATION OF (+)-CATECHIN, (-)-EPICATECHIN, (-)-CATECHIN, (+)-EPICATECHIN, AND THEIR 5,7,3',4'-TETRA-O-BENZYL ANALOGUES MARS, INCORPORATED (US) 2008-03-12 EP claimed
WO-2007002877-A1 PREPARATION OF (+)-CATECHIN, (-)-EPICATECHIN, (-)-CATECHIN, (+)-EPICATECHIN, AND THEIR 5,7,3',4'-TETRA-O-BENZYL ANALOGUES MARS, INCORPORATED (US) 2007-01-04 WO claimed
EP-2822653-B1 NEW C-GLYCOSYLPOLYPHENOL ANTIDIABETIC AGENTS, EFFECT ON GLUCOSE TOLERANCE AND INTERACTION WITH BETA-AMYLOID. THERAPEUTIC APPLICATIONS OF THE SYNTHESIZED AGENT(S) AND OF GENISTA TENERA ETHYL ACETATE EXTRACTS CONTAINING SOME OF THOSE AGENTS FACULDADE DE CIENCIAS DA UNIV DE LISBOA (PT) 2024-06-19 EP disclosed
CN-117794526-A Compositions and methods for antioxidants and anti-inflammatory therapeutics 阿万蒂生物科学股份有限公司 2024-03-29 CN disclosed
CN-113710262-B Scutellaria baicalensis composition and method for taste modulation 国际香料和香精公司 2024-01-05 CN disclosed
US-20230053152-A1 Novel Quercetin Redox Derivative And Use Thereof As BET Inhibitor BENOBIO CO., LTD. (KR) 2023-02-16 US disclosed
WO-2023288020-A1 COMPOSITIONS AND METHODS FOR ANTIOXIDANT AND ANTI-INFLAMMATORY THERAPEUTICS AVANTI BIOSCIENCES INC. (US) 2023-01-19 WO disclosed
CN-113710262-A Scutellaria baicalensis composition and method for taste modulation 国际香料和香精公司 2021-11-26 CN disclosed
CN-112724114-A Epicatechin and related polyphenols 斯法尔制药私人有限公司 2021-04-30 CN disclosed
EP-2981260-B1 NOVEL ANALOGUES OF EPICATECHIN AND RELATED POLYPHENOLS SPHAERA PHARMA PRIVATE LTD (IN) 2021-01-13 EP disclosed
US-20040029914-A1 Novel flavanoids as chemotherapeutic, chemopreventive, and antiangiogenic agents SRI INTERNATIONAL 2004-02-12 US disclosed
US-20030229136-A1 Novel flavanoids as chemotherapeutic, chemopreventive, and antiangiogenic agents SRI INTERNATIONAL 2003-12-11 US disclosed
WO-2003089423-A2 NOVEL FLAVANOIDS AND CHALCONES AS CHEMOTHERAPEUTIC, CHEMOPREVENTIVE, AND ANTIANGIOGENIC AGENTS SRI INTERNATIONAL (US) 2003-10-30 WO disclosed
US-4348333-A β-Ketocarboxyl and phosphonate dihydro-chalcone sweeteners THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1982-09-07 US disclosed
US-4290957-A SWEETENERS DYNAPOL (US) 1981-09-22 US disclosed
US-4283434-A FOR FOODS NUTRASWEET COMPANY THE 1981-08-11 US disclosed
US-4267165-A Comestibles sweetened with alpha amino acid dihydrochalcones DYNAPOL (US) 1981-05-12 US disclosed
US-4226804-A ARTIFICIAL SWEETENER DYNAPOL (US) 1980-10-07 US disclosed
US-4204007-A 4-(Dihydroxyhexoxy)dihydrochalcone sweeteners DYNAPOL (US) 1980-05-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040029914-A1 Novel flavanoids as chemotherapeutic, chemopreventive, and antiangiogenic agents FLT1, VEGFA, FLT4 MAOB 1380/4885MEN1 3385/4885KMT2A 3690/4885
US-20030229136-A1 Novel flavanoids as chemotherapeutic, chemopreventive, and antiangiogenic agents FLT1, VEGFA, FLT4 MAOB 1370/4885MEN1 3434/4885KMT2A 3666/4885
US-20100048920-A1 Preparation of (+)-Catechin, (-)-Epicatechin, (-)-Catechin, and (+)-Epicatechin and Their 5,7,3',4'-Tetra-O-Benzyl Analogues HAAO, TES, HPD MAOB 882/4885MEN1 4540/4885KMT2A 2842/4885
US-20230053152-A1 Novel Quercetin Redox Derivative And Use Thereof As BET Inhibitor BET1, BRD4, BRD3 MAOB 1784/4885MEN1 4278/4885KMT2A 884/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.