SCHEMBL6581696

SCHEMBL6581696

Cc1ccc(-c2nc(-c3cccc(C(C)(C)N)c3)n(C)n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 4/20 0.51
NR1H3 Q13133 4/20 0.51
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
HSD17B2 P37059 1/20 0.48
TMEM97 Q5BJF2 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
NMT1 P30419 1/20 0.42
ADORA2A P29274 2/20 0.42
ADORA1 P30542 2/20 0.42
TDP2 O95551 4/20 0.41
SIRT1 Q96EB6 1/20 0.41
KDM4C Q9H3R0 2/20 0.41
AKT1 P31749 1/20 0.38
AKT2 P31751 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17279740 0.75 NR1H3 (0.82) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL6581144 0.75 NR1H2 (0.53) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL6581290 0.73 NR1H2 (0.50) NR1H2NR1H3NPC1RAB9AHSD17B2
Hydrochloric Acid SCHEMBL6580743 0.72 NR1H2 (0.49) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL822566 0.69 NR1H3 (1.00) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL25599752 0.69 NR1H2 (0.71) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL22307346 0.69 NR1H3 (0.82) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL3910446 0.67 ACHE (0.50) CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL11557551 0.67 NPC1 (0.57) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL6915245 0.67 KDM4E (0.48) TMEM97SIGMAR1SMN1; SMN2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP claimed