SCHEMBL6581144

SCHEMBL6581144

Cc1ccc(-c2nc(-c3cccc(C=O)c3)n(C)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 4/20 0.53
NR1H3 Q13133 4/20 0.53
NPC1 O15118 4/20 0.53
RAB9A P51151 4/20 0.53
HSD17B2 P37059 1/20 0.49
TDP2 O95551 3/20 0.45
SIRT1 Q96EB6 1/20 0.45
KDM4C Q9H3R0 2/20 0.45
TRIM24 O15164 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
BRD4 O60885 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
ADORA2A P29274 2/20 0.40
ADORA1 P30542 2/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
MEN1 O00255 2/20 0.39
POLB P06746 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6580839 0.87 KDM4C (0.49) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL6581289 0.83 DRD1 (0.46) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL6578166 0.82 HSD17B2 (0.51) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL6580847 0.80 TDP2 (0.44) NR1H2NR1H3NPC1RAB9AHSD17B2
Pyrrolidine SCHEMBL6582654 0.80 KDM4C (0.43) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL17279740 0.76 NR1H3 (0.82) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL2321575 0.76 TRIM24 (0.61) NPC1RAB9ATRIM24TRIM33BRD4
SCHEMBL30249928 0.76 TRIM24 (0.61) NPC1RAB9ATRIM24TRIM33BRD4
SCHEMBL6581696 0.75 NR1H2 (0.51) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL6581290 0.74 NR1H2 (0.50) NR1H2NR1H3NPC1RAB9AHSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1148357-C Triazole and imidazole derivative - 2004-05-05 CN disclosed
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
CN-1281852-A Triazole and imidazole derivative HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed