SCHEMBL6582793

SCHEMBL6582793

COc1ccc(-c2nc(-c3cccc(C=O)c3)nn2CC2CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.47
NR1H3 Q13133 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.43
PTGIR P43119 1/20 0.42
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
AVPR1B P47901 8/20 0.39
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
TDP2 O95551 1/20 0.38
TSHR P16473 1/20 0.37
CRHR1 P34998 1/20 0.37
AXL P30530 1/20 0.36
TYRO3 Q06418 1/20 0.36
MERTK Q12866 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582750 0.97 NR1H2 (0.46) NR1H2NR1H3L3MBTL1PTGIRNPC1
SCHEMBL6582832 0.96 L3MBTL1 (0.43) NR1H2NR1H3L3MBTL1PTGIRAVPR1B
SCHEMBL6581016 0.93 AVPR1B (0.43) NR1H2NR1H3L3MBTL1PTGIRAVPR1B
SCHEMBL6584155 0.86 NR1H3 (0.51) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6578548 0.84 NR1H3 (0.64) NR1H2NR1H3L3MBTL1NPC1RAB9A
SCHEMBL6578958 0.83 NR1H3 (0.48) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6584100 0.83 NR1H2 (0.48) NR1H2NR1H3L3MBTL1NPC1RAB9A
SCHEMBL6584148 0.83 NR1H3 (0.48) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6581065 0.83 NR1H3 (0.48) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6580723 0.82 NR1H2 (0.47) NR1H2NR1H3NPC1RAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed