SCHEMBL6583033

SCHEMBL6583033

COc1cc(CCCC2NC(=O)OC2=O)ccc1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
TAAR1 Q96RJ0 2/20 0.48
MAPK1 P28482 2/20 0.48
TSHR P16473 2/20 0.48
LMNA P02545 1/20 0.47
GLA P06280 1/20 0.47
CALM1 P0DP23 1/20 0.46
ALOX5 P09917 2/20 0.46
OR51E2 Q9H255 1/20 0.46
PTPN1 P18031 2/20 0.46
SHBG P04278 3/20 0.46
CYP3A4 P08684 3/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP2C8 P10632 1/20 0.44
CYP2B6 P20813 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581977 0.96 MTNR1A (0.47) MTNR1AMTNR1BTAAR1MAPK1TSHR
SCHEMBL6581895 0.93 TAAR1 (0.50) MTNR1AMTNR1BTAAR1MAPK1TSHR
SCHEMBL8889117 0.88 GAA (0.42) MTNR1AMTNR1BTSHRALDH1A1GAA
SCHEMBL6583757 0.86 TNKS2 (0.43) ALOX5CYP3A4GAAMET
SCHEMBL6584139 0.83 CYP3A4 (0.49) TSHRLMNACYP3A4CYP1A2GAA
SCHEMBL6583581 0.83 SMN1; SMN2 (0.42) MAPK1TSHRLMNAALDH1A1GAA
SCHEMBL6583798 0.81 GAA (0.44) TSHRALDH1A1GAATDP1
SCHEMBL8334676 0.79 MTNR1A (0.51) MTNR1AMTNR1BTAAR1MAPK1TSHR
SCHEMBL7165617 0.78 ESR1 (0.38) TAAR1LMNACALM1SHBGCYP3A4
SCHEMBL6584720 0.77 MTNR1A (0.52) MTNR1AMTNR1BCYP3A4CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0710659-B1 Oxazolidinedione derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-01-28 EP disclosed
WO-1997000249-A1 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-03 WO disclosed
EP-0710659-A1 Oxazolidinedione derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-08 EP disclosed