SCHEMBL6583633

SCHEMBL6583633

O=C(Nc1ccc(Oc2ccnc(NCCc3ccccc3)n2)c2ccccc12)NC1CC1C1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 20/20 0.45
MAPK14 Q16539 5/20 0.45
SRC P12931 8/20 0.40
SYK P43405 8/20 0.40
HCK P08631 1/20 0.39
GSK3B P49841 1/20 0.39
MAPK12 P53778 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6587587 0.89 SYK (0.44) GSK3AMAPK14SRCSYKHCK
SCHEMBL6583148 0.88 GSK3A (0.42) GSK3AMAPK14SRCSYKHCK
SCHEMBL6584730 0.86 GSK3A (0.43) GSK3AMAPK14SRCSYKHCK
SCHEMBL6583161 0.83 GSK3A (0.42) GSK3AMAPK14SRCSYKHCK
SCHEMBL6585819 0.83 KDR (0.40) GSK3AMAPK14SRCSYKHCK
SCHEMBL6585714 0.82 KDR (0.44) GSK3AMAPK14SRCSYKMAPK12
SCHEMBL6583630 0.80 MAPK14 (0.40) GSK3AMAPK14SRCSYKHCK
SCHEMBL6581723 0.78 SYK (0.38) GSK3AMAPK14SRCSYK
SCHEMBL6585511 0.76 VCP (0.39) GSK3AMAPK14SRCSYKHCK
SCHEMBL6598212 0.76 KDR (0.40) GSK3AMAPK14SRCSYKHCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004534787-A 2004-11-18 JP claimed
EP-1414810-A2 1,4-DISUBSTITUTED BENZO-FUSED CYCLOALKYL UREA COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-05-06 EP claimed
WO-2002098869-A2 1,4-DISUBSTITUTED BENZO-FUSED CYCLOALKYL UREA COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-12 WO claimed