SCHEMBL6584477

SCHEMBL6584477

N#Cc1ccccc1S(=O)(=O)n1ccc2cccc(N3CCNCC3)c21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 18/20 0.49
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
CYP1A2 P05177 1/20 0.41
HTR1A P08908 1/20 0.41
CYP2D6 P10635 1/20 0.41
NCF1 P14598 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
HTR2A P28223 1/20 0.41
HTR7 P34969 1/20 0.41
MTOR P42345 1/20 0.41
HTR3A P46098 1/20 0.41
HTR5A P47898 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SIGMAR1 Q99720 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202033 0.80 HTR6 (0.66) HTR6CYP1A2HTR1AHTR1BHTR2A
Hydrochloric Acid SCHEMBL5201694 0.79 HTR6 (0.65) HTR6CYP1A2HTR1AHTR1BHTR2A
SCHEMBL6585144 0.75 HTR6 (0.60) HTR6CYP1A2HTR1AHTR1BHTR2A
SCHEMBL6589771 0.72 HTR6 (0.61) HTR6HTR3EHTR3BCYP1A2HTR1A
SCHEMBL233169 0.72 ADRB1 (0.58) HTR6HTR3EHTR3BCYP1A2HTR1A
SCHEMBL3621241 0.72 HTR6 (0.50) HTR6HTR2AKDM4EALDH1A1
Hydrochloric Acid SCHEMBL29882725 0.71 ADRB1 (0.56) HTR6HTR3EHTR3BCYP1A2HTR1A
Hydrochloric Acid SCHEMBL20139829 0.71 ADRB1 (0.56) HTR6HTR3EHTR3BCYP1A2HTR1A
SCHEMBL5483901 0.70 HTR6 (0.74) HTR6
SCHEMBL1136474 0.70 HTR6 (0.76) HTR6HTR3EHTR3BCYP1A2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414442-A1 3-ARYLSULFONYL-7-PIPERAZINYL- INDOLES, -BENZOFURANS AND -BENZOTHIOPHENES WITH 5-HT6 RECEPTOR AFFINITY FOR TREATING CNS DISORDERS SMITHKLINE BEECHAM PLC (GB) 2004-05-06 EP claimed
WO-2003013510-A1 3-ARYLSULFONYL-7-PIPERAZINYL- INDOLES, -BENZOFURANS AND -BENZOTHIOPHENES WITH 5-HT6 RECEPTOR AFFINITY FOR TREATING CNS DISORDERS SMITHKLINE BEECHAM P.L.C. (GB) 2003-02-20 WO claimed