SCHEMBL6585855

SCHEMBL6585855

CC1(C)C(=O)Nc2c(OCCCN3CCCN(Cc4ccc5ccccc5n4)CC3)cccc21

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.41
HTR7 P34969 1/20 0.41
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
FAAH O00519 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
DRD2 P14416 3/20 0.38
HCRTR1 O43613 5/20 0.38
HCRTR2 O43614 5/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581869 0.97 HTR1A (0.43) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL6583402 0.95 HTR1A (0.43) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL8310206 0.89 HTR1A (0.42) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL6584265 0.88 HTR1A (0.40) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL6583227 0.85 HTR1A (0.44) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL8309662 0.85 HTR1A (0.40) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL6585292 0.85 HTR1A (0.42) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL6581635 0.85 HTR1A (0.40) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL6588676 0.83 DRD2 (0.47) DRD2
SCHEMBL6585787 0.83 MEN1 (0.43) HTR1AHTR7MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957100-B1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME KOWA CO (JP) 2004-10-27 EP disclosed
EP-0957100-A1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME Kowa Co., Ltd. (JP) 1999-11-17 EP disclosed