SCHEMBL6586253

SCHEMBL6586253

CCC(C)c1cc(-c2nc3c(OC(N)=O)cccc3[nH]2)on1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 16/20 0.38
HPSE Q9Y251 1/20 0.36
PKN1 Q16512 1/20 0.36
PKN2 Q16513 1/20 0.36
CBFB Q13951 1/20 0.35
PLA2G2A P14555 1/20 0.34
ALOX15 P16050 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6804664 0.85 PARP1 (0.51) PARP1PKN1PKN2
SCHEMBL6589472 0.83 PKN2 (0.39) PARP1HPSEPKN1PKN2PLA2G2A
SCHEMBL6587689 0.82 PARP1 (0.39) PARP1HPSECBFBPLA2G2AALOX15
SCHEMBL6591556 0.80 PARP1 (0.40) PARP1HPSEPKN1PKN2PLA2G2A
SCHEMBL6586846 0.78 PARP1 (0.46) PARP1
SCHEMBL6591532 0.75 PARP1 (0.41) PARP1HPSEPLA2G2AALOX15PTGS2
SCHEMBL6589114 0.74 PARP1 (0.57) PARP1HPSEPKN1PKN2CBFB
SCHEMBL6591503 0.73 PARP1 (0.44) PARP1HPSEPKN1PKN2PLA2G2A
SCHEMBL6804675 0.73 PARP1 (0.36) PARP1PKN1PKN2
SCHEMBL6591536 0.72 PARP1 (0.39) PARP1HPSECBFBPLA2G2AALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed