SCHEMBL6586303

SCHEMBL6586303

COc1ccccc1Oc1c(Cl)nc(N2CCOCC2)nc1C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
LMNA P02545 2/20 0.43
HSD17B10 Q99714 2/20 0.43
POLB P06746 1/20 0.43
GPR55 Q9Y2T6 1/20 0.43
KDM4E B2RXH2 2/20 0.42
MAPT P10636 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
MEN1 O00255 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
AGER Q15109 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALDH1A1 P00352 1/20 0.42
EDNRB P24530 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5631503 0.88 MAPT (0.49) HTTLMNAHSD17B10POLBKDM4E
SCHEMBL4065446 0.85 PIK3CA (0.51) HTTLMNAHSD17B10POLBGPR55
SCHEMBL6586305 0.84 DHPS (0.55) LMNAHSD17B10KDM4EMAPTTDP1
SCHEMBL4068802 0.83 DHPS (0.50) EDNRBEDNRADHPS
SCHEMBL7841637 0.80 EDNRB (0.54) EDNRBEDNRA
SCHEMBL5633057 0.78 MAPT (0.49) LMNAHSD17B10POLBKDM4EMAPT
SCHEMBL5653603 0.77 EDNRB (0.65) EDNRBEDNRA
SCHEMBL7850537 0.77 EDNRA (0.49) HTTKDM4EMAPTL3MBTL1MEN1
SCHEMBL7990192 0.77 PIK3CA (0.36) HTTLMNAHSD17B10POLBGPR55
SCHEMBL5764886 0.75 EDNRB (0.53) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0897914-B1 Process for the preparation of 2,5-disubstitued pyridines HOFFMANN LA ROCHE (CH) 2004-05-26 EP claimed
WO-2002083650-A1 NOVEL SULFONYLAMINO-PYRIMIDINES ACTELION PHARMACEUTICALS LTD (CH) 2002-10-24 WO disclosed