SCHEMBL6586376

SCHEMBL6586376

O=C(O)c1nc2c(OCc3ccccc3)cccc2[nH]c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 2/20 0.52
DHODH Q02127 7/20 0.50
DRD2 P14416 2/20 0.45
DRD4 P21917 2/20 0.45
DRD3 P35462 2/20 0.45
PDE5A O76074 1/20 0.44
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
FOLH1 Q04609 1/20 0.44
SRD5A1 P18405 1/20 0.43
ADORA3 P0DMS8 1/20 0.42
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6079636 0.86 GABRA1 (0.56) SRD5A2DHODHDRD2DRD4DRD3
SCHEMBL9528101 0.76 RHEB (0.55) SRD5A2DHODHDRD2DRD4DRD3
SCHEMBL7619109 0.76 DRD2 (0.67) SRD5A2DHODHDRD2DRD4DRD3
SCHEMBL6080461 0.75 FOLH1 (0.50) SRD5A2FOLH1MRGPRX4LMNA
SCHEMBL20597759 0.75 SRD5A2 (0.48) SRD5A2DHODHDRD2DRD4DRD3
SCHEMBL6081154 0.74 GRIN1 (0.45) DHODHLMNA
SCHEMBL18304068 0.74 DRD2 (0.51) SRD5A2DHODHDRD2DRD4DRD3
SCHEMBL9527738 0.74 PDE5A (0.51) SRD5A2DHODHDRD2DRD4DRD3
SCHEMBL27629254 0.73 MRGPRX4 (0.55) SRD5A2FOLH1MRGPRX4
SCHEMBL5619518 0.72 DHODH (0.79) DHODHPDE5APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP claimed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO claimed
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed