SCHEMBL6587116

SCHEMBL6587116

COc1ccc(C2=CC(N)(C(=O)C(C)(C)c3ccc4ccccc4c3)N=N2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.37
RAB9A P51151 5/20 0.37
CASP3 P42574 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
PARP1 P09874 2/20 0.35
ALOX5 P09917 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2A6 P11509 1/20 0.34
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 3/20 0.34
NFKB1 P19838 2/20 0.34
NFKB2 Q00653 2/20 0.34
RELA Q04206 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 2/20 0.34
HPGD P15428 2/20 0.34
GABBR2 O75899 1/20 0.34
GABBR1 Q9UBS5 1/20 0.34
LMNA P02545 1/20 0.34
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581999 0.69 CSNK2A2 (0.57) NPC1RAB9ALMNA
SCHEMBL6585131 0.69 MTNR1A (0.46) ALDH1A1MAPTHPGDL3MBTL1MMP9
SCHEMBL7890086 0.67 HTT (0.43) NPC1RAB9AALDH1A1KDM4ESMN1; SMN2
SCHEMBL17295890 0.64 CYP1A2 (0.55) NPC1RAB9ACASP3SENP7CYP1A2
SCHEMBL19149202 0.64 CYP1A2 (0.55) NPC1RAB9ACASP3SENP7CYP1A2
SCHEMBL6438107 0.63 CYP1A2 (0.57) NPC1RAB9ACASP3SENP7CYP1A2
SCHEMBL27941075 0.63 MAPT (0.58) ALDH1A1KDM4EMAPTGAA
SCHEMBL14580025 0.62 CYP1A2 (0.49) NPC1RAB9ACASP3SENP7CYP1A2
SCHEMBL4678770 0.62 PTPN1 (0.49) MAPT
SCHEMBL505821 0.62 AKR1C3 (0.55) CYP1A2CYP2A6ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945440-B1 AMINOPYRAZOLE DERIVATIVES BANYU PHARMA CO LTD (JP) 2004-05-26 EP claimed