SCHEMBL6587178

SCHEMBL6587178

NC(=O)Oc1cccc2[nH]c(-c3ccn(-c4ccc(Cl)cc4[N+](=O)[O-])c3)nc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.41
CHEK2 O96017 1/20 0.40
PKN1 Q16512 1/20 0.38
PKN2 Q16513 1/20 0.38
NPBWR1 P48145 1/20 0.34
GRIK1 P39086 1/20 0.34
GRIA1 P42261 1/20 0.34
GRIA2 P42262 1/20 0.34
GRIA3 P42263 1/20 0.34
GRIA4 P48058 1/20 0.34
GRIK2 Q13002 1/20 0.34
GRIK3 Q13003 1/20 0.34
GRIK4 Q16099 1/20 0.34
GRIK5 Q16478 1/20 0.34
HPSE Q9Y251 1/20 0.34
GAA P10253 3/20 0.33
MGAM O43451 2/20 0.33
SI P14410 2/20 0.33
MGAM2 Q2M2H8 2/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6806378 0.87 PARP1 (0.57) PARP1CHEK2PKN1PKN2
SCHEMBL7480129 0.83 MGAM (0.52) PARP1PKN1PKN2NPBWR1HPSE
SCHEMBL6587289 0.82 PARP1 (0.49) PARP1CHEK2PKN1PKN2HPSE
SCHEMBL6588648 0.81 PARP1 (0.40) PARP1CHEK2PKN1PKN2HPSE
SCHEMBL6806385 0.77 CHEK2 (0.40) PARP1CHEK2NPBWR1GRIK1GRIA1
SCHEMBL6587399 0.75 HPSE (0.42) PARP1HPSEGAAMGAMSI
SCHEMBL6591184 0.74 AURKB (0.44) PARP1CHEK2PKN1PKN2HPSE
SCHEMBL6586096 0.73 PARP1 (0.53) PARP1CHEK2PKN1PKN2HPSE
SCHEMBL6588713 0.71 HPSE (0.43) PARP1CHEK2PKN1PKN2HPSE
SCHEMBL6591596 0.70 PARP1 (0.48) PARP1CHEK2PKN1PKN2HPSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed