SCHEMBL6587399

SCHEMBL6587399

Cc1cccc(C)c1-n1ccc(-c2nc3c(OC(N)=O)cccc3[nH]2)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPSE Q9Y251 2/20 0.42
PARP1 P09874 12/20 0.41
MGAM O43451 5/20 0.41
GAA P10253 5/20 0.41
SI P14410 5/20 0.41
MGAM2 Q2M2H8 5/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PLA2G2A P14555 1/20 0.40
ALOX15 P16050 1/20 0.40
PTGS2 P35354 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6807298 0.84 PARP1 (0.60) PARP1PLA2G2AALOX15PTGS2
SCHEMBL6586096 0.83 PARP1 (0.53) HPSEPARP1PLA2G2AALOX15PTGS2
SCHEMBL6587289 0.82 PARP1 (0.49) HPSEPARP1MGAMGAASI
SCHEMBL6591184 0.82 AURKB (0.44) HPSEPARP1PLA2G2AALOX15PTGS2
SCHEMBL6588713 0.81 HPSE (0.43) HPSEPARP1PLA2G2AALOX15PTGS2
SCHEMBL6588648 0.80 PARP1 (0.40) HPSEPARP1PLA2G2AALOX15PTGS2
SCHEMBL6587303 0.76 EPHX2 (0.52) HPSEPARP1PLA2G2AALOX15PTGS2
SCHEMBL6586851 0.76 PIM1 (0.48) HPSEPARP1KDM4EALDH1A1HPGD
SCHEMBL6589916 0.76 TUBB4A (0.44) HPSEPARP1TP53
SCHEMBL6578530 0.75 PARP1 (0.67) HPSEPARP1KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed