SCHEMBL6587439

SCHEMBL6587439

CC(C)CCCN1CCC(OC(=O)C(O)(c2ccccc2)C2CCC2)CC1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.64
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
HTT P42858 1/20 0.55
CHRM3 P20309 4/20 0.53
CHRM2 P08172 2/20 0.53
CHRM4 P08173 1/20 0.53
CHRM5 P08912 1/20 0.53
CHRM1 P11229 1/20 0.53
HRH1 P35367 1/20 0.53
HTR2B P41595 1/20 0.53
KCNH2 Q12809 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7649694 0.82 ALDH1A1 (0.82) ALDH1A1CYP1A2CYP3A4CYP2D6CHRM3
SCHEMBL6589129 0.82 CHRM2 (0.66) ALDH1A1CYP1A2CYP3A4CYP2D6HTT
SCHEMBL6587556 0.82 CHRM2 (0.66) CHRM3CHRM2CHRM1
SCHEMBL5544972 0.81 ALDH1A1 (0.75) ALDH1A1CYP1A2CYP3A4CYP2D6HTT
SCHEMBL5542878 0.81 ALDH1A1 (0.75) ALDH1A1CYP1A2CYP3A4CYP2D6HTT
SCHEMBL4298699 0.80 ALDH1A1 (0.86) ALDH1A1CYP1A2CYP3A4CYP2D6HTT
SCHEMBL28075363 0.80 ALDH1A1 (0.59) ALDH1A1CYP1A2CYP3A4CYP2D6HTT
SCHEMBL29409726 0.79 ALDH1A1 (0.84) ALDH1A1CYP1A2CYP3A4CYP2D6HTT
SCHEMBL6589592 0.79 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4CYP2D6HTT
SCHEMBL1697179 0.78 ALDH1A1 (1.00) ALDH1A1CYP1A2CYP3A4CYP2D6HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823423-B1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMA CO LTD (JP) 2004-06-16 EP claimed
CN-1188471-A 1,4-disubstituted piepridine derivatives BANYU PHARMA CO LTD (JP) 1998-07-22 CN claimed
EP-0823423-A1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1998-02-11 EP claimed
EP-0823423-B1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMA CO LTD (JP) 2004-06-16 EP disclosed
CN-1188471-A 1,4-disubstituted piepridine derivatives BANYU PHARMA CO LTD (JP) 1998-07-22 CN disclosed
US-5750540-A SIDE EFFECT REDUCTION BANYU PHARMACEUTICAL CO., LTD. (JP) 1998-05-12 US disclosed
EP-0823423-A1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1998-02-11 EP disclosed