SCHEMBL6587744

SCHEMBL6587744

CCc1nc(-c2nc3c(OC(N)=O)cccc3[nH]2)c[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 2/20 0.44
PARP1 P09874 13/20 0.42
ALOX15 P16050 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HPSE Q9Y251 2/20 0.39
PLA2G2A P14555 1/20 0.38
PTGS2 P35354 1/20 0.38
PIM1 P11309 2/20 0.37
GSK3A P49840 2/20 0.37
DYRK1A Q13627 2/20 0.37
PIM3 Q86V86 2/20 0.37
AURKB Q96GD4 2/20 0.37
CLK4 Q9HAZ1 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6810500 0.83 PARP1 (0.56) PARP1ALOX15PLA2G2APTGS2PIM1
SCHEMBL6585207 0.81 PARP1 (0.51) CBFBPARP1ALOX15ALDH1A1TP53
SCHEMBL6585540 0.78 CBFB (0.47) CBFBPARP1ALOX15ALDH1A1TP53
SCHEMBL6585381 0.75 CBFB (0.67) CBFBPARP1ALOX15ALDH1A1TP53
SCHEMBL6591546 0.74 PARP1 (0.44) PARP1ALOX15HPSEPLA2G2APTGS2
SCHEMBL7479706 0.74 PARP1 (0.49) PARP1ALOX15HPSEPLA2G2APTGS2
SCHEMBL6590890 0.74 METAP2 (0.50) CBFBPARP1ALOX15ALDH1A1TP53
SCHEMBL6588173 0.74 PARP1 (0.49) PARP1ALDH1A1HPSEPIM1
SCHEMBL6384512 0.73 PARP1 (0.56) PARP1ALOX15HPSEPLA2G2APTGS2
SCHEMBL6586775 0.73 PARP1 (0.46) PARP1ALOX15HPSEPLA2G2APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed