SCHEMBL6587787

SCHEMBL6587787

NC(=O)Oc1cccc2[nH]c(-c3cnccc3OCCCN3CCN(Cc4ccccc4)CC3)nc12

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.46
AURKB Q96GD4 2/20 0.46
KDR P35968 1/20 0.46
PARP1 P09874 10/20 0.42
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 3/20 0.42
POLB P06746 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
USP2 O75604 1/20 0.42
TDP1 Q9NUW8 1/20 0.40
DRD2 P14416 1/20 0.38
HTR6 P50406 1/20 0.38
DHODH Q02127 2/20 0.38
HTR1A P08908 2/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584782 0.96 AURKA (0.46) AURKAAURKBKDRPARP1ALDH1A1
SCHEMBL6587697 0.90 AURKB (0.44) AURKAAURKBKDRPARP1ALDH1A1
SCHEMBL6590117 0.90 PARP1 (0.51) AURKAAURKBPARP1ALDH1A1KDM4E
SCHEMBL6806120 0.90 AURKB (0.58) AURKAAURKBKDRPARP1DHODH
SCHEMBL6589815 0.89 PARP1 (0.52) AURKAAURKBPARP1ALDH1A1KDM4E
SCHEMBL6587227 0.89 PARP1 (0.44) AURKAAURKBKDRPARP1ALDH1A1
SCHEMBL6583719 0.86 PARP1 (0.43) AURKAAURKBKDRPARP1ALDH1A1
SCHEMBL6587192 0.86 PARP1 (0.50) AURKBPARP1KDM4EDHODHHTR1A
SCHEMBL6802857 0.85 AURKB (0.59) AURKAAURKBKDRPARP1DHODH
SCHEMBL6587212 0.85 AURKA (0.50) AURKAAURKBKDRPARP1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed