SCHEMBL6587227

SCHEMBL6587227

NC(=O)Oc1cccc2[nH]c(-c3cnccc3OCCCN3CCNCC3)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.44
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
DHODH Q02127 1/20 0.39
AURKB Q96GD4 4/20 0.39
AURKA O14965 2/20 0.39
MKNK2 Q9HBH9 3/20 0.37
PIM1 P11309 2/20 0.37
PIM3 Q86V86 2/20 0.37
PRKD3 O94806 1/20 0.37
SRC P12931 1/20 0.37
FLT4 P35916 1/20 0.37
KDR P35968 1/20 0.37
CLK2 P49760 1/20 0.37
GSK3A P49840 1/20 0.37
DYRK1A Q13627 1/20 0.37
PRKD2 Q9BZL6 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
STK17A Q9UEE5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7534102 0.96 PARP1 (0.43) PARP1ALDH1A1KDM4ETDP1DHODH
SCHEMBL6590117 0.93 PARP1 (0.51) PARP1ALDH1A1KDM4EDHODHAURKB
SCHEMBL6589815 0.92 PARP1 (0.52) PARP1ALDH1A1KDM4EDHODHAURKB
SCHEMBL6587697 0.92 AURKB (0.44) PARP1ALDH1A1KDM4EDHODHAURKB
SCHEMBL6799952 0.89 PARP1 (0.56) PARP1DHODHAURKBAURKAMKNK2
SCHEMBL6587192 0.89 PARP1 (0.50) PARP1KDM4EDHODHAURKBMKNK2
SCHEMBL6587787 0.89 AURKA (0.46) PARP1ALDH1A1KDM4ETDP1DHODH
SCHEMBL6583586 0.88 PARP1 (0.51) PARP1ALDH1A1KDM4EDHODHAURKB
SCHEMBL6583719 0.87 PARP1 (0.43) PARP1ALDH1A1KDM4EDHODHAURKB
SCHEMBL6806003 0.84 PARP1 (0.56) PARP1DHODHAURKBAURKAMKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed