SCHEMBL6589047

SCHEMBL6589047

NC(=O)Oc1cccc2[nH]c(-c3c(Br)cnn3Cc3ccc(Cl)cc3)nc12

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.41
TSHR P16473 1/20 0.38
PTGDR2 Q9Y5Y4 3/20 0.36
GRM2 Q14416 1/20 0.36
GAA P10253 2/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MGAM O43451 1/20 0.35
SI P14410 1/20 0.35
MGAM2 Q2M2H8 1/20 0.35
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6805077 0.86 PARP1 (0.58) PARP1TSHR
SCHEMBL6805083 0.75 TSHR (0.48) PARP1TSHRPTGDR2GRM2SMN1; SMN2
SCHEMBL7763612 0.74 PARP1 (0.41) PARP1GAALMNASMN1; SMN2L3MBTL1
SCHEMBL6585205 0.74 PARP1 (0.42) PARP1GRM2GAALMNASMN1; SMN2
SCHEMBL6591596 0.73 PARP1 (0.48) PARP1GAAMGAMSIMGAM2
SCHEMBL6591702 0.72 PARP1 (0.44) PARP1GAALMNASMN1; SMN2L3MBTL1
SCHEMBL6384512 0.71 PARP1 (0.56) PARP1
SCHEMBL6383679 0.71 PARP1 (0.72) PARP1
SCHEMBL6587289 0.70 PARP1 (0.49) PARP1GAAMGAMSIMGAM2
SCHEMBL6381152 0.70 PARP1 (0.73) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed