SCHEMBL6805083

SCHEMBL6805083

NC(=O)c1cccc2nc(-c3c(Br)cnn3Cc3ccc(Cl)cc3)[nH]c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
PARP1 P09874 9/20 0.40
PLK4 O00444 1/20 0.37
CHEK1 O14757 1/20 0.37
AURKA O14965 1/20 0.37
DAPK3 O43293 1/20 0.37
MAP4K4 O95819 1/20 0.37
CSF1R P07333 1/20 0.37
RET P07949 1/20 0.37
FGFR1 P11362 1/20 0.37
PDGFRA P16234 1/20 0.37
LTK P29376 1/20 0.37
KDR P35968 1/20 0.37
MAP2K2 P36507 1/20 0.37
FLT3 P36888 1/20 0.37
CSNK1A1 P48729 1/20 0.37
PRKX P51817 1/20 0.37
CDK5 Q00535 1/20 0.37
MAP2K1 Q02750 1/20 0.37
MST1R Q04912 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6805077 0.85 PARP1 (0.58) TSHRPARP1PLK4MAP4K4PRKX
SCHEMBL6589047 0.75 PARP1 (0.41) TSHRPARP1GRM2SMN1; SMN2PTGDR2
SCHEMBL6806912 0.73 GRM2 (0.44) PARP1FGFR1GRM2PARP2PARP3
SCHEMBL6810614 0.72 MAP4K4 (0.52) PARP1PLK4CHEK1AURKADAPK3
SCHEMBL6807085 0.72 NR3C2 (0.43) PARP1PLK4CHEK1AURKADAPK3
SCHEMBL6807111 0.69 PARP1 (0.46) PARP1PLK4MAP4K4KDRPRKX
SCHEMBL6810628 0.69 PARP1 (0.52) PARP1PARP2PARP3
SCHEMBL6804457 0.69 PARP1 (0.42) PARP1PARP2PARP3KMT2ASMN1; SMN2
SCHEMBL6804448 0.68 GRM2 (0.38) PARP1FGFR1BTKCD38GRM2
SCHEMBL7138977 0.67 PARP1 (0.50) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed