SCHEMBL6589453

SCHEMBL6589453

O=C(Cl)c1scc(CCl)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.41
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
GPR35 Q9HC97 1/20 0.31
F10 P00742 1/20 0.30
KEAP1 Q14145 1/20 0.30
NFE2L2 Q16236 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6587977 0.78 KMT2A (0.39) GSK3BKDM4EGAAF10
SCHEMBL2722085 0.71 F10 (0.41) GSK3BKDM4EGAAGPR35F10
SCHEMBL11236244 0.69
SCHEMBL6596838 0.68 GPR35 (0.42) GSK3BKDM4EGAAGPR35KEAP1
SCHEMBL4078686 0.68 GPR35 (0.42) GSK3BKDM4EGAAGPR35KEAP1
SCHEMBL13887939 0.68 GSK3B (0.38) GSK3BKDM4EGAAF10
SCHEMBL6594590 0.67 CYP2A6 (0.36) KDM4EGPR35
SCHEMBL1279064 0.65 KDM4E (0.45) KDM4EGAAF10
SCHEMBL11325227 0.64 GPR35 (0.39) GSK3BGPR35
SCHEMBL3814347 0.64 KDM4E (0.52) KDM4EGAAF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1143855-C I (ortho)-anthranilamide derivatives as anti-coagulants ���ֹɷݹ�˾ 2004-03-31 CN disclosed
EP-1040108-B1 ORTHO-ANTHRANILAMIDE DERIVATIVES AS ANTI-COAGULANTS SCHERING AG (DE) 2004-02-25 EP disclosed
US-6498185-B1 ENZYME FACTOR XA INHIBITORS BERLEX LABORATORIES, INC. 2002-12-24 US disclosed
US-6380221-B1 FOR THERAPY OF DISEASE-STATES CHARACTERIZED BY THROMBOTIC ACTIVITY BERLEX LABORATORIES, INC. 2002-04-30 US disclosed
CN-1282329-A I (ortho)-anthranilamide derivatives as anti-coagulants SCHERING AG (DE) 2001-01-31 CN disclosed
US-6140351-A FOR TREATING THROMBOSIS BERLEX LABORATORIES, INC. (US) 2000-10-31 US disclosed
EP-1040108-A1 ORTHO-ANTHRANILAMIDE DERIVATIVES AS ANTI-COAGULANTS SCHERING AKTIENGESELLSCHAFT (DE) 2000-10-04 EP disclosed
WO-1999032477-A1 ORTHO-ANTHRANILAMIDE DERIVATIVES AS ANTI-COAGULANTS SCHERING AKTIENGESELLSCHAFT (DE) 1999-07-01 WO disclosed