SCHEMBL6589568

SCHEMBL6589568

Cc1nc(Sc2ccc(F)cc2)cc(Sc2ccc(F)cc2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
ALDH1A1 P00352 6/20 0.43
LMNA P02545 4/20 0.43
HPGD P15428 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
NPSR1 Q6W5P4 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ATM Q13315 2/20 0.41
HTT P42858 2/20 0.40
TP53 P04637 1/20 0.39
CYP1A2 P05177 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP3A4 P08684 1/20 0.37
NOTUM Q6P988 1/20 0.36
TYMS P04818 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27418234 0.81 MEN1 (0.44) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL576260 0.75 MEN1 (0.48) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL7938033 0.73 ACHE (0.68) MAPTMEN1KMT2AALDH1A1L3MBTL1
SCHEMBL20408990 0.69 KMT2A (0.40) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL8736568 0.69 NPC1 (0.44) MAPTMEN1KMT2ALMNAL3MBTL1
SCHEMBL7937262 0.69 MEN1 (0.55) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL31669638 0.69 MEN1 (0.50) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL3451400 0.69 MEN1 (0.61) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL13812416 0.68 MAPT (0.46) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL755938 0.68 MEN1 (0.39) MAPTMEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0781766-B1 HETEROCYCLIC DERIVATIVE AND MEDICINE NIPPON SHINYAKU CO LTD (JP) 2004-03-31 EP disclosed
US-6191149-B1 DRUG FOR CEREBROVASCULAR DISEASE NIPPON SHINYAKU, CO., LTD. (JP) 2001-02-20 US disclosed
US-5945426-A PREVENT NEURONAL DEATH NIPPON SHINYAKU CO., LTD. (JP) 1999-08-31 US disclosed
EP-0781766-A1 HETEROCYCLIC DERIVATIVE AND MEDICINE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1997-07-02 EP disclosed