SCHEMBL6590308

SCHEMBL6590308

O=C(O)c1cc(O)c2cc(-c3ccco3)cc(OCc3ccccc3)c2n1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PPARD Q03181 4/20 0.40
MCL1 Q07820 2/20 0.40
XDH P47989 1/20 0.40
MAP4K4 O95819 1/20 0.40
PTPN1 P18031 2/20 0.39
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6079995 0.90 HPGD (0.44) MAPTKDM4EALDH1A1HPGDTSHR
SCHEMBL6594732 0.81 MCL1 (0.49) MCL1XDHMAP4K4PTPN1
SCHEMBL6080055 0.81 POLB (0.47) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL6592298 0.80 MCL1 (0.53) MAPTPPARDMCL1MAP4K4PTPN1
SCHEMBL6588409 0.80 MCL1 (0.46) MCL1XDHMAP4K4PTPN1
SCHEMBL6593585 0.80 CYP11B1 (0.47) MAPTMCL1MAP4K4PTPN1
SCHEMBL6595828 0.80 MRGPRX4 (0.44) MCL1MAP4K4PTPN1
SCHEMBL6594866 0.79 PTGER1 (0.44) MAPTHPGDSMN1; SMN2MCL1XDH
SCHEMBL6080208 0.79 PTGER1 (0.47) MCL1
SCHEMBL6080497 0.78 MRGPRX4 (0.51) MCL1XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP claimed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO claimed
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed