SCHEMBL6592298

SCHEMBL6592298

COc1ccc(-c2cc(OCc3ccccc3)c3nc(C(=O)O)cc(O)c3c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 8/20 0.53
MAPT P10636 3/20 0.46
NPSR1 Q6W5P4 2/20 0.46
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
PTPN1 P18031 2/20 0.45
MAPK1 P28482 2/20 0.45
NOD2 Q9HC29 1/20 0.45
PPARD Q03181 1/20 0.44
MAP4K4 O95819 1/20 0.44
DHODH Q02127 1/20 0.44
ANO1 Q5XXA6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080550 0.92 MAPT (0.45) MCL1MAPTNPSR1CTSLCTSB
SCHEMBL6594732 0.88 MCL1 (0.49) MCL1PTPN1MAP4K4
SCHEMBL6591608 0.86 MCL1 (0.51) MCL1MAPTMAPK1
SCHEMBL6588409 0.84 MCL1 (0.46) MCL1PTPN1MAP4K4DHODH
SCHEMBL6595828 0.84 MRGPRX4 (0.44) MCL1PTPN1MAP4K4DHODH
SCHEMBL6080319 0.82 CNR1 (0.46) MCL1MAPTPTPN1PPARDMAP4K4
SCHEMBL6593585 0.82 CYP11B1 (0.47) MCL1MAPTPTPN1MAP4K4
SCHEMBL6595262 0.81 ALOX15 (0.51) MCL1DHODH
SCHEMBL6079891 0.81 MCL1 (0.53) MCL1MAPTNPSR1MAPK1
SCHEMBL6590308 0.80 MAPT (0.42) MCL1MAPTPTPN1PPARDMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed