SCHEMBL6590849

SCHEMBL6590849

C[C@@H](CC(N)=O)CC(=O)N(CC1SC=CC1=O)C1CCCNCC1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.33
SLC6A4 P31645 12/20 0.33
SLC6A3 Q01959 6/20 0.33
CYP2D6 P10635 2/20 0.33
KCNH2 Q12809 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6595138 0.72 SLC6A4 (0.32) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL4768429 0.71 SLC6A2 (0.38) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL7023360 0.65 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL6593956 0.64 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3
SCHEMBL4767101 0.63 CTSD (0.37) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL6591070 0.63
SCHEMBL4765027 0.61 CTSD (0.45) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL4768444 0.60
SCHEMBL6589463 0.59
SCHEMBL6587495 0.59 TRPM8 (0.35) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP claimed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP claimed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO claimed
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed