SCHEMBL659146

SCHEMBL659146

O=C(O)CC(Cc1nc2ccc(Oc3ccccc3)cc2[nH]1)c1ccc(Cl)cc1

nearest known ligand 0.73

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRKCZ Q05513 9/20 0.73
FNTA P49354 3/20 0.47
FNTB P49356 3/20 0.47
EGLN2 Q96KS0 1/20 0.47
EGLN1 Q9GZT9 1/20 0.47
RAB9A P51151 1/20 0.47
GRIN1 Q05586 3/20 0.46
GRIN2B Q13224 3/20 0.46
PIN1 Q13526 1/20 0.45
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
CHEK2 O96017 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL659145 0.92 PRKCZ (0.64) PRKCZFNTAFNTBEGLN2EGLN1
Hydrochloric Acid SCHEMBL658866 0.91 PRKCZ (0.63) PRKCZFNTAFNTBEGLN2EGLN1
SCHEMBL657824 0.91 PRKCZ (0.60) PRKCZRAB9AGRIN1GRIN2BPIN1
SCHEMBL2303038 0.88 PRKCZ (0.72) PRKCZFNTAFNTBEGLN1GRIN1
SCHEMBL659484 0.86 PRKCZ (0.83) PRKCZRAB9APIN1
SCHEMBL10252755 0.85 PRKCZ (0.78) PRKCZRAB9APIN1
SCHEMBL2304303 0.85 PRKCZ (0.78) PRKCZRAB9APIN1
SCHEMBL2301693 0.85 PRKCZ (1.00) PRKCZRAB9APIN1CHEK2
SCHEMBL2302990 0.84 PRKCZ (0.76) PRKCZRAB9APIN1
SCHEMBL2303682 0.83 PRKCZ (0.90) PRKCZRAB9APIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349999-A1 ALLOSTERIC PROTEIN KINASE MODULATORS Universität des Saarlandes (DE) 2011-08-03 EP claimed
WO-2010043711-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2010-04-22 WO claimed
EP-2349999-B1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIV SAARLAND (DE) 2016-01-27 EP disclosed
EP-2349999-B1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIV SAARLAND (DE) 2016-01-27 EP disclosed
US-8912186-B2 Allosteric protein kinase modulators UNIVERSITAET DES SAARLANDES (DE) 2014-12-16 US disclosed
US-8912186-B2 Allosteric protein kinase modulators UNIVERSITAET DES SAARLANDES (DE) 2014-12-16 US disclosed
US-8912186-B2 Allosteric protein kinase modulators UNIVERSITAET DES SAARLANDES (DE) 2014-12-16 US disclosed
US-20120046307-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2012-02-23 US disclosed
US-20120046307-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2012-02-23 US disclosed
US-20120046307-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2012-02-23 US disclosed
EP-2349999-A1 ALLOSTERIC PROTEIN KINASE MODULATORS Universität des Saarlandes (DE) 2011-08-03 EP disclosed
WO-2010043711-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2010-04-22 WO disclosed
WO-2010043711-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2010-04-22 WO disclosed
EP-2177510-A1 Allosteric protein kinase modulators Universität des Saarlandes (DE) 2010-04-21 EP disclosed
EP-2177510-A1 Allosteric protein kinase modulators Universität des Saarlandes (DE) 2010-04-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046307-A1 ALLOSTERIC PROTEIN KINASE MODULATORS AURKC, AURKA, AURKB PRKCZ 26/4885FNTA 944/4885FNTB 1890/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.