SCHEMBL6592099

SCHEMBL6592099

Cc1ccc(NC(=O)c2sc3ccccc3c2Cl)c(C(=O)Nc2cccnc2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
F10 P00742 19/20 1.00
NPC1 O15118 1/20 0.73
LMNA P02545 1/20 0.73
RAB9A P51151 1/20 0.73
SMN1; SMN2 Q16637 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590511 0.89 F10 (1.00) F10SMN1; SMN2
SCHEMBL6594123 0.87 F10 (0.89) F10SMN1; SMN2
SCHEMBL29865482 0.86 MAPT (0.74) F10NPC1LMNARAB9ASMN1; SMN2
SCHEMBL23353332 0.86 MAPT (0.74) F10NPC1LMNARAB9ASMN1; SMN2
SCHEMBL6593805 0.85 F10 (1.00) F10
SCHEMBL6591396 0.85 F10 (1.00) F10
SCHEMBL16384127 0.85 RAB9A (1.00) F10NPC1LMNARAB9ASMN1; SMN2
SCHEMBL6591720 0.84 F10 (0.82) F10
SCHEMBL6592241 0.83 F10 (1.00) F10SMN1; SMN2
SCHEMBL6592119 0.83 F10 (1.00) F10NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040108-B1 ORTHO-ANTHRANILAMIDE DERIVATIVES AS ANTI-COAGULANTS SCHERING AG (DE) 2004-02-25 EP claimed
US-6380221-B1 FOR THERAPY OF DISEASE-STATES CHARACTERIZED BY THROMBOTIC ACTIVITY BERLEX LABORATORIES, INC. 2002-04-30 US claimed
EP-1040108-B1 ORTHO-ANTHRANILAMIDE DERIVATIVES AS ANTI-COAGULANTS SCHERING AG (DE) 2004-02-25 EP disclosed
US-6498185-B1 ENZYME FACTOR XA INHIBITORS BERLEX LABORATORIES, INC. 2002-12-24 US disclosed
US-6380221-B1 FOR THERAPY OF DISEASE-STATES CHARACTERIZED BY THROMBOTIC ACTIVITY BERLEX LABORATORIES, INC. 2002-04-30 US disclosed
US-6140351-A FOR TREATING THROMBOSIS BERLEX LABORATORIES, INC. (US) 2000-10-31 US disclosed