SCHEMBL6592136

SCHEMBL6592136

Cc1[nH]cnc1-c1nc2c(OC(N)=O)cccc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.43
HPSE Q9Y251 2/20 0.41
ALOX15 P16050 2/20 0.39
CBFB Q13951 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PLA2G2A P14555 1/20 0.39
PTGS2 P35354 1/20 0.39
PKN1 Q16512 1/20 0.38
PKN2 Q16513 1/20 0.38
DHODH Q02127 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6805344 0.82 PARP1 (0.59) PARP1ALOX15PLA2G2APTGS2PKN1
SCHEMBL6585540 0.77 CBFB (0.47) PARP1HPSEALOX15CBFBALDH1A1
SCHEMBL6587182 0.77 MEN1 (0.52) PARP1HPSEALOX15CBFBALDH1A1
SCHEMBL6585182 0.76 PARP1 (0.47) PARP1HPSEALOX15PLA2G2APTGS2
SCHEMBL6591546 0.76 PARP1 (0.44) PARP1HPSEALOX15PLA2G2APTGS2
SCHEMBL6591503 0.75 PARP1 (0.44) PARP1HPSEALOX15ALDH1A1TP53
SCHEMBL7479706 0.75 PARP1 (0.49) PARP1HPSEALOX15PLA2G2APTGS2
SCHEMBL7471031 0.75 PARP1 (0.45) PARP1HPSEALDH1A1CYP3A4CYP2C19
SCHEMBL6585381 0.75 CBFB (0.67) PARP1ALOX15CBFBALDH1A1TP53
SCHEMBL7827732 0.74 PARP1 (0.69) PARP1HPSEALOX15PLA2G2APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed