SCHEMBL6596743

SCHEMBL6596743

CCc1ccc(C2=CC(C)(C)Sc3ccc(C#Cc4ccc(C(=O)O)cn4)cc32)cc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.49
CYP26A1 O43174 1/20 0.49
RARA P10276 14/20 0.49
RARB P10826 14/20 0.49
RARG P13631 14/20 0.49
KMT2A Q03164 1/20 0.44
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
EGLN1 Q9GZT9 1/20 0.35
GRM5 P41594 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6591838 0.91 RARA (0.56) CYP3A4CYP26A1RARARARBRARG
SCHEMBL6590791 0.90 RARA (0.53) CYP3A4CYP26A1RARARARBRARG
SCHEMBL726359 0.89 RARA (0.60) CYP3A4CYP26A1RARARARBRARG
SCHEMBL6593885 0.84 RARA (0.57) CYP3A4CYP26A1RARARARBRARG
SCHEMBL1140748 0.81 RARA (0.48) CYP3A4RARARARBRARGKMT2A
SCHEMBL1140826 0.80 RARB (0.60) RARARARBRARGKMT2ANPC1
SCHEMBL6589951 0.78 RARA (0.64) CYP3A4CYP26A1RARARARBRARG
SCHEMBL14384928 0.78 RARB (0.53) RARARARBRARGKMT2ANPC1
SCHEMBL6587152 0.77 RARB (0.56) CYP3A4CYP26A1RARARARBRARG
SCHEMBL13784637 0.77 RARA (0.42) RARARARBRARGSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042313-B1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY ALLERGAN INC (US) 2004-04-28 EP disclosed
EP-1042313-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY Allergan Sales, Inc. (US) 2000-10-11 EP disclosed
WO-1999033821-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST-LIKE ACTIVITY ALLERGAN SALES, INC. (US) 1999-07-08 WO disclosed