SCHEMBL6598291

SCHEMBL6598291

CN(C)c1ncnc2ccc([NH])cc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 14/20 0.59
CYP3A4 P08684 13/20 0.59
CLK4 Q9HAZ1 12/20 0.59
ALDH1A1 P00352 10/20 0.59
LMNA P02545 10/20 0.59
MAPK1 P28482 8/20 0.59
HSD17B10 Q99714 3/20 0.59
MEN1 O00255 1/20 0.59
TP53 P04637 1/20 0.59
CASP1 P29466 1/20 0.59
CASP7 P55210 1/20 0.59
KMT2A Q03164 1/20 0.59
CYP2D6 P10635 8/20 0.54
CYP2C19 P33261 7/20 0.54
TSHR P16473 7/20 0.54
CYP2C9 P11712 3/20 0.54
HIF1A Q16665 5/20 0.52
USP2 O75604 3/20 0.51
GLA P06280 1/20 0.51
HPGD P15428 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31031351 0.80 CYP1A2 (0.61) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL2998447 0.79 EGFR (0.68) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL4357581 0.79 ALDH1A1 (0.69) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL25844376 0.79 CYP1A2 (0.59) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL31031354 0.75 CYP1A2 (0.55) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL2880252 0.75 CYP1A2 (0.55) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL4359084 0.73 CYP1A2 (0.75) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL4353312 0.73 CYP1A2 (0.75) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL2184445 0.73 EGFR (0.68) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL2993744 0.72 IRAK4 (0.53) CYP1A2CYP3A4CLK4ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1373252-A1 CHEMICAL DERIVATIVES AND THEIR USE AS ANTI-TELOMERASE AGENT Aventis Pharma S.A. (FR) 2004-01-02 EP disclosed
WO-2002076975-A1 CHEMICAL DERIVATIVES AND THEIR USE AS ANTI-TELOMERASE AGENT AVENTIS PHARMA S.A. (FR) 2002-10-03 WO disclosed