SCHEMBL6598927

SCHEMBL6598927

Cc1nn(-c2cccc3cnccc23)cc1OC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.38
DRD2 P14416 3/20 0.38
DRD3 P35462 3/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPKAPK2 P49137 1/20 0.38
HTR1A P08908 2/20 0.37
DRD4 P21917 2/20 0.37
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
TRPV1 Q8NER1 3/20 0.36
SLC22A12 Q96S37 1/20 0.36
ALDH1A1 P00352 2/20 0.36
NR3C1 P04150 1/20 0.36
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
NPY5R Q15761 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
KCNA3 P22001 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6312276 0.82 HTR2C (0.47) HTR2CKDM4EMAPKAPK2OPRM1OPRL1
SCHEMBL6599323 0.79 SLC22A12 (0.40) HTR2CKDM4EMAPKAPK2OPRM1OPRL1
SCHEMBL1680249 0.75 NPC1 (0.45) ALDH1A1MEN1MAPK1KMT2ACYP3A4
SCHEMBL6319301 0.75 HTR2C (0.43) HTR2CKDM4EMAPKAPK2TRPV1MEN1
SCHEMBL6261873 0.74 HTR2C (0.42) HTR2CKDM4EMAPKAPK2OPRM1ALDH1A1
Hydrochloric Acid SCHEMBL6313986 0.74 HTR2C (0.43) HTR2CKDM4EMAPKAPK2TRPV1MEN1
Hydrochloric Acid SCHEMBL6313991 0.73 HTR2C (0.42) HTR2CKDM4EMAPKAPK2OPRM1ALDH1A1
SCHEMBL6313000 0.73 L3MBTL1 (0.44) HTR2CKDM4ETRPV1ALDH1A1MAPK1
SCHEMBL6312111 0.71 KDM4E (0.49) HTR2CKDM4EMAPKAPK2OPRM1OPRL1
SCHEMBL19187423 0.69 MAPT (0.47) HTR2CDRD2DRD3KDM4EMAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056729-B1 N-[(SUBSTITUTED FIVE-MEMBERED DI- OR TRIAZA DIUNSATURATED RING)CARBONYL]GUANIDINE DERIVATIVES FOR THE TREATMENT OF ISCHEMIA PFIZER PROD INC (US) 2004-12-29 EP claimed