SCHEMBL6599243

SCHEMBL6599243

COc1c(C(=O)O)n(Cc2ccc(Cl)c(Cl)c2)c2ccc(O)cc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 4/20 1.00
CCR2 P41597 16/20 0.76
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083775 0.88 ABCB11 (0.78) ABCB11CCR2ALDH1A1GAAMAPT
SCHEMBL6599266 0.87 ABCB11 (0.77) ABCB11CCR2ALDH1A1GAAMAPT
SCHEMBL6598122 0.85 ABCB11 (0.74) ABCB11CCR2ALDH1A1GAAMAPT
SCHEMBL6599182 0.85 ABCB11 (0.73) ABCB11CCR2
SCHEMBL6781272 0.83 ABCB11 (0.71) ABCB11CCR2
SCHEMBL21465476 0.81 ABCB11 (0.68) ABCB11CCR2ALDH1A1MAPTPKM
SCHEMBL21465479 0.80 ABCB11 (0.67) ABCB11CCR2ALDH1A1MAPTPKM
SCHEMBL6780182 0.80 ABCB11 (0.66) ABCB11CCR2
SCHEMBL5213205 0.79 ABCB11 (0.66) ABCB11CCR2ALDH1A1MAPTPKM
SCHEMBL5212313 0.77 ABCB11 (0.62) ABCB11CCR2ALDH1A1MAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150952-B1 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2004-10-27 EP disclosed
US-6737435-B1 ANTIINFLAMMATORY AGENTS; MONOCYTE CHEMOATTRACTANT PROTEIN-1 (MCP-1) DISEASES ASTRAZENECA AB (SE) 2004-05-18 US disclosed