SCHEMBL6600429

SCHEMBL6600429

CS(=O)(=O)OCC1CN(c2ccc(C(=N)NC(=O)c3cccnc3)cc2)C(=O)O1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 4/20 0.40
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
NAE1 Q13564 1/20 0.38
UBA3 Q8TBC4 1/20 0.38
ITGB3 P05106 4/20 0.37
PRSS1 P07477 4/20 0.37
PRSS2 P07478 4/20 0.37
ITGA2B P08514 4/20 0.37
PRSS3 P35030 4/20 0.37
F10 P00742 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
TP53 P04637 1/20 0.36
ABCB11 O95342 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601789 0.89 GRM2 (0.45) GRM2ITGB3PRSS1PRSS2ITGA2B
SCHEMBL6600722 0.89 GRM2 (0.45) GRM2ITGB3PRSS1PRSS2ITGA2B
SCHEMBL6600718 0.89 GRM2 (0.45) GRM2ITGB3PRSS1PRSS2ITGA2B
SCHEMBL7631925 0.89 ITGB3 (0.53) GRM2ITGB3PRSS1PRSS2ITGA2B
SCHEMBL7638635 0.88 ITGB3 (0.48) ITGB3PRSS1PRSS2ITGA2BPRSS3
SCHEMBL7640299 0.88 ITGB3 (0.43) ALDH1A1TSHRITGB3ITGA2BF10
SCHEMBL7640396 0.87 ITGB3 (0.43) ITGB3PRSS1PRSS2ITGA2BPRSS3
SCHEMBL7639718 0.87 ITGB3 (0.39) ALDH1A1TSHRITGB3PRSS1PRSS2
SCHEMBL7640285 0.86 ITGB3 (0.42) ITGB3PRSS1PRSS2ITGA2BPRSS3
SCHEMBL7633585 0.86 ITGB3 (0.38) ALDH1A1TSHRITGB3PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2004-01-28 EP disclosed
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed