SCHEMBL7640299

SCHEMBL7640299

CC(C)OC(=O)CN1CCN(CC2CN(c3ccc(C(=N)NC(=O)c4cccnc4)cc3)C(=O)O2)CC1.CS(=O)(=O)OCC1CN(c2ccc(C(=N)NC(=O)c3cccnc3)cc2)C(=O)O1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
ALDH1A1 P00352 2/20 0.34
TSHR P16473 1/20 0.34
SIGMAR1 Q99720 5/20 0.34
ACACB O00763 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
F10 P00742 1/20 0.33
PTGDR Q13258 1/20 0.33
HTR7 P34969 1/20 0.33
SORT1 Q99523 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
MAPT P10636 2/20 0.33
MAPK1 P28482 1/20 0.33
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6600840 0.93 ITGB3 (0.48) ITGB3ITGA2BSIGMAR1ACACBSMN1; SMN2
SCHEMBL7633208 0.93 ITGB3 (0.45) ITGB3ITGA2BALDH1A1SIGMAR1SMN1; SMN2
SCHEMBL7631925 0.91 ITGB3 (0.53) ITGB3ITGA2BSIGMAR1F10
SCHEMBL7639718 0.91 ITGB3 (0.39) ITGB3ITGA2BALDH1A1TSHRSIGMAR1
SCHEMBL7633507 0.89 ITGB3 (0.49) ITGB3ITGA2BALDH1A1SIGMAR1SMN1; SMN2
SCHEMBL7640427 0.88 ITGB3 (0.43) ITGB3ITGA2BALDH1A1SIGMAR1F10
SCHEMBL6600429 0.88 GRM2 (0.40) ITGB3ITGA2BALDH1A1TSHRSMN1; SMN2
SCHEMBL7637805 0.87 ITGB3 (0.43) ITGB3ITGA2BALDH1A1SIGMAR1SMN1; SMN2
SCHEMBL7640396 0.87 ITGB3 (0.43) ITGB3ITGA2BSIGMAR1ACACBF10
SCHEMBL7639664 0.86 ITGB3 (0.44) ITGB3ITGA2BSIGMAR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6455529-B1 OXAZOLIDIN-2-ONE DERIVATIVES; ANTICOAGULANTS; ANTIMETASTASIS, ANTICARCINOGENIC, ANTIISCHEMIC, AND ANTIINFLAMMATORY AGENTS; OSTEOPOROSIS, ARTERIOSCLEROSIS MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2002-09-24 US disclosed