SCHEMBL6600529

SCHEMBL6600529

Fc1ccc(-c2[nH]cnc2-c2cccc(Br)n2)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 10/20 0.54
MAPK13 O15264 3/20 0.54
MAPK12 P53778 3/20 0.54
MAPK11 Q15759 3/20 0.54
RAF1 P04049 1/20 0.54
MAPK9 P45984 1/20 0.54
BRD4 O60885 1/20 0.46
IDO1 P14902 5/20 0.46
CYP3A4 P08684 3/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
NR3C2 P08235 1/20 0.41
MAPK10 P53779 1/20 0.40
TGFBR1 P36897 1/20 0.39
TGFBR2 P37173 1/20 0.39
TNIK Q9UKE5 1/20 0.39
GSK3B P49841 1/20 0.39
GCGR P47871 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6808551 0.79 MAPK14 (0.60) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL15571062 0.77 ALDH1A1 (0.43) CYP3A4KDM4EMAPTTGFBR1
SCHEMBL10992179 0.77 MAPK14 (0.83) MAPK14MAPK13MAPK12MAPK11RAF1
Hydrochloric Acid SCHEMBL30023185 0.76 MAPK14 (0.80) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL11967202 0.75 MAPK14 (0.56) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL6599716 0.75 SNCA (0.46) MAPK14MAPK13MAPK12MAPK11CYP3A4
Pyrimidine SCHEMBL6804171 0.72 MAPK14 (0.47) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL4536537 0.71 MAPK14 (0.66) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL4434902 0.70 MAPK14 (1.00) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL6423292 0.70 MAPK14 (1.00) MAPK14MAPK13MAPK12MAPK11RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349851-A4 COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-09-08 EP disclosed
EP-1349851-A1 COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2003-10-08 EP disclosed
WO-2002040468-A1 COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2002-05-23 WO disclosed