SCHEMBL6600536

SCHEMBL6600536

NC(=O)c1noc(C(Cc2ccc3ccccc3c2)N(C(N)=O)C(=O)[CH]Cc2ccc3ccccc3c2)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A11 Q9UPY5 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
PSMB5 P28074 1/20 0.32
EPHX1 P07099 1/20 0.32
MMP9 P14780 1/20 0.31
MMP8 P22894 1/20 0.31
MC5R P33032 4/20 0.31
MC4R P32245 2/20 0.31
MC3R P41968 2/20 0.31
DPP4 P27487 1/20 0.31
OPRM1 P35372 1/20 0.31
MC1R Q01726 2/20 0.31
FCER2 P06734 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CTRB1 P17538 1/20 0.31
GHSR Q92847 1/20 0.30
PPARG P37231 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601730 0.90 ZAP70 (0.34) SLC7A11HTR2AHTR2CHTR2BPSMB5
SCHEMBL6601217 0.89 PSMB5 (0.36) SLC7A11HTR2AHTR2CHTR2BPSMB5
SCHEMBL3728180 0.87 SLC7A11 (0.35) SLC7A11PSMB5MMP9MMP8FCER2
SCHEMBL6600950 0.87 CAPN1 (0.37) SLC7A11FCER2GHSR
SCHEMBL6601080 0.86 SMN1; SMN2 (0.38) FCER2MEN1KMT2A
SCHEMBL6600540 0.77 MC4R (0.42) SLC7A11HTR2AHTR2CHTR2BEPHX1
SCHEMBL4284133 0.76 MAOB (0.37) SLC7A11PSMB5MMP9MMP8GHSR
SCHEMBL6606297 0.75 PSMB5 (0.37) SLC7A11HTR2AHTR2CHTR2BPSMB5
SCHEMBL6600426 0.75 CAPN1 (0.39) SLC7A11FCER2PPARGPPARDPPARA
SCHEMBL4282444 0.74 CAPN1 (0.39) PSMB5MMP9MMP8FCER2GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805816-B1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK AS (DK) 2004-07-28 EP claimed
EP-0805816-B1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK AS (DK) 2004-07-28 EP disclosed
US-6350767-B1 GROWTH HORMONE RELEASE STIMULANT NOVO NORDISK A/S (DK) 2002-02-26 US disclosed
US-6013658-A ANIMAL GROWTH REGULATORS NOVO NORDISK A/S (DK) 2000-01-11 US disclosed
EP-0907374-A1 GROWTH HORMONE COMPONENT AND BONE ANTI-RESORPTIVE AGENT IN CYCLIC (COHERENCE) TREATMENT OF OSTEOPOROSIS NOVO NORDISK A/S (DK) 1999-04-14 EP disclosed
WO-1997046252-A1 GROWTH HORMONE COMPONENT AND BONE ANTI-RESORPTIVE AGENT IN CYCLIC (COHERENCE) TREATMENT OF OSTEOPOROSIS NOVO NORDISK A/S (DK) 1997-12-11 WO disclosed
EP-0805816-A1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK A/S (DK) 1997-11-12 EP disclosed
WO-1996022997-A1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK A/S (DK) 1996-08-01 WO disclosed