SCHEMBL6600939

SCHEMBL6600939

CCCCOC(=O)CCN1CCN(CC2CN(c3ccc(C(=N)NC(=O)OC)cc3)C(=O)O2)CC1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.50
ITGA2B P08514 6/20 0.50
GRM2 Q14416 2/20 0.48
SIGMAR1 Q99720 12/20 0.43
PRSS1 P07477 4/20 0.41
PRSS2 P07478 4/20 0.41
PRSS3 P35030 4/20 0.41
F10 P00742 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6600829 0.92 ITGB3 (0.45) ITGB3ITGA2BGRM2SIGMAR1PRSS1
SCHEMBL6601660 0.92 ITGB3 (0.59) ITGB3ITGA2BGRM2SIGMAR1PRSS1
SCHEMBL6601266 0.92 ITGB3 (0.59) ITGB3ITGA2BGRM2SIGMAR1PRSS1
SCHEMBL6601938 0.91 ITGB3 (0.44) ITGB3ITGA2BGRM2SIGMAR1PRSS1
SCHEMBL6600978 0.91 ITGB3 (0.46) ITGB3ITGA2BGRM2SIGMAR1PRSS1
SCHEMBL6599465 0.90 ITGB3 (0.51) ITGB3ITGA2BGRM2SIGMAR1PRSS1
SCHEMBL6603429 0.90 ITGB3 (0.46) ITGB3ITGA2BGRM2SIGMAR1PRSS1
SCHEMBL6601365 0.89 ITGB3 (0.47) ITGB3ITGA2BGRM2SIGMAR1PRSS1
SCHEMBL6601257 0.89 ITGB3 (0.44) ITGB3ITGA2BGRM2SIGMAR1PRSS1
SCHEMBL6603381 0.88 ITGB3 (0.44) ITGB3ITGA2BGRM2SIGMAR1PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2004-01-28 EP disclosed
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed