SCHEMBL6601119

SCHEMBL6601119

COC(=O)CN1CCN(CC2CN(c3ccc(C(=N)NC(=O)c4cccnc4)cc3)C(=O)O2)CC1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.52
ITGA2B P08514 1/20 0.52
SIGMAR1 Q99720 12/20 0.42
GRM2 Q14416 1/20 0.40
F10 P00742 1/20 0.39
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601597 0.93 ITGB3 (0.60) ITGB3ITGA2BSIGMAR1GRM2F10
SCHEMBL6600840 0.92 ITGB3 (0.48) ITGB3ITGA2BSIGMAR1GRM2F10
SCHEMBL6602428 0.92 ITGB3 (0.45) ITGB3ITGA2BSIGMAR1GRM2ADRA2A
SCHEMBL6602652 0.91 ITGB3 (0.55) ITGB3ITGA2BSIGMAR1GRM2F10
SCHEMBL6605657 0.90 ITGB3 (0.51) ITGB3ITGA2BSIGMAR1GRM2
SCHEMBL6602405 0.89 ITGB3 (0.48) ITGB3ITGA2BSIGMAR1GRM2F10
SCHEMBL6602426 0.88 ITGB3 (0.46) ITGB3ITGA2BSIGMAR1GRM2F10
SCHEMBL6599782 0.87 ITGB3 (0.51) ITGB3ITGA2BSIGMAR1GRM2F10
SCHEMBL7631925 0.86 ITGB3 (0.53) ITGB3ITGA2BSIGMAR1GRM2F10
SCHEMBL6602820 0.86 ITGB3 (0.59) ITGB3ITGA2BSIGMAR1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2004-01-28 EP disclosed
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed