SCHEMBL6601480

SCHEMBL6601480

Cc1cc(C)cc(C(=O)N2CC2C)c1.Cc1cc(C)cc(C(=O)O)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.59
ALDH1A1 P00352 2/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HTT P42858 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
HCAR1 Q9BXC0 1/20 0.47
HPGD P15428 2/20 0.46
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
CNR2 P34972 1/20 0.39
TP53 P04637 2/20 0.39
TACR1 P25103 2/20 0.38
HCAR2 Q8TDS4 1/20 0.38
GAA P10253 2/20 0.37
MAPT P10636 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3890994 0.93 ALDH1A1 (0.59) TPMTALDH1A1NPSR1HTTL3MBTL1
SCHEMBL2823144 0.82 DHODH (0.51) ALDH1A1HTTL3MBTL1RXRARXRB
SCHEMBL6918093 0.79 TPMT (0.94) TPMTALDH1A1HCAR1HPGDRXRA
SCHEMBL221684 0.77 TPMT (1.00) TPMTALDH1A1HCAR1HPGDRXRA
SCHEMBL3898423 0.76 HTT (0.76) HTTL3MBTL1HPGDLMNANPC1
SCHEMBL27894302 0.76 L3MBTL1 (0.55) ALDH1A1HTTL3MBTL1HPGDGAA
SCHEMBL6918090 0.74 TPMT (0.94) TPMTALDH1A1HCAR1HPGDRXRA
SCHEMBL6914123 0.74 TPMT (0.94) TPMTALDH1A1HCAR1HPGDRXRA
SCHEMBL6916035 0.74 TPMT (0.94) TPMTALDH1A1HCAR1HPGDRXRA
SCHEMBL6918621 0.74 TPMT (0.94) TPMTALDH1A1HCAR1HPGDRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402900-A1 MEDICINAL COMPOSITIONS Takeda Chemical Industries, Ltd. (JP) 2004-03-31 EP disclosed
EP-1354603-A1 CONCOMITANT DRUGS Takeda Chemical Industries, Ltd. (JP) 2003-10-22 EP disclosed