SCHEMBL6601767

SCHEMBL6601767

CCCCCCN1CCCC(COc2ccc(C(=O)c3c(-c4ccc(OC)cc4)sc4cc(OC)ccc34)cc2)C1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 17/20 0.63
ESR2 Q92731 17/20 0.63
ENPP3 O14638 2/20 0.54
ENPP1 P22413 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601833 0.92 ESR1 (0.63) ESR1ESR2
SCHEMBL6604899 0.88 ESR1 (0.67) ESR1ESR2ENPP3ENPP1
SCHEMBL6601884 0.84 ESR1 (0.61) ESR1ESR2ENPP3ENPP1
SCHEMBL6959934 0.83 ESR1 (0.86) ESR1ESR2ENPP3ENPP1
SCHEMBL7665997 0.83 ESR1 (0.86) ESR1ESR2ENPP3ENPP1
SCHEMBL7663013 0.83 ESR1 (0.86) ESR1ESR2ENPP3ENPP1
SCHEMBL7664893 0.83 ESR1 (0.86) ESR1ESR2ENPP3ENPP1
SCHEMBL6601387 0.83 ESR1 (0.64) ESR1ESR2ENPP3ENPP1
SCHEMBL8492628 0.83 CHRNB2 (0.55) ESR1ESR2
SCHEMBL7671368 0.82 ESR1 (0.88) ESR1ESR2ENPP3ENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0905132-B1 Benzothiophenes LILLY CO ELI (US) 2004-08-04 EP disclosed
US-6060488-A ANTICARCINOGENIC AGENTS; POSTMENOPAUSAL CANCER OF BREASTS, UTERUS, CERVIX ELI LILLY AND COMPANY (US) 2000-05-09 US disclosed
EP-0905132-A1 Benzothiophenes ELI LILLY AND COMPANY (US) 1999-03-31 EP disclosed