SCHEMBL6601912

SCHEMBL6601912

CCCCC#Cc1cccc2c(OCc3ccccc3)cc(C(=O)O)nc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
PTGER1 P34995 4/20 0.39
MRGPRX4 Q96LA9 3/20 0.39
XDH P47989 1/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
APEX1 P27695 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ALOX15 P16050 1/20 0.37
MCL1 Q07820 1/20 0.37
PTGES O14684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6079882 0.92 CTSL (0.46) CTSLCTSBMRGPRX4KDM4ELMNA
SCHEMBL6596521 0.89 XDH (0.40) CTSLCTSBPTGER1XDHKDM4E
SCHEMBL6596257 0.88 CTSL (0.43) CTSLCTSBPTGER1MRGPRX4XDH
SCHEMBL6594101 0.83 MCL1 (0.43) PTGER1MRGPRX4XDHALOX15MCL1
SCHEMBL6080213 0.82 CTSL (0.44) CTSLCTSBXDHKDM4ELMNA
SCHEMBL6079887 0.80 KDM4E (0.37) CTSLCTSBKDM4ELMNACYP1A2
SCHEMBL6080269 0.80 CTSL (0.48) CTSLCTSBMRGPRX4KDM4ELMNA
SCHEMBL6591127 0.78 MRGPRX4 (0.40) PTGER1MRGPRX4XDHMCL1
SCHEMBL6079765 0.76 NOTUM (0.41) MRGPRX4LMNAMAPTHSD17B10TDP1
SCHEMBL6590520 0.75 MRGPRX4 (0.47) PTGER1MRGPRX4CYP1A2MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP claimed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO claimed
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed