SCHEMBL6602154

SCHEMBL6602154

CCC(=O)CC(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.62
GSK3B P49841 2/20 0.58
MMP1 P03956 1/20 0.54
CES2 O00748 1/20 0.52
CES1 P23141 1/20 0.52
HDAC1 Q13547 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
MMP2 P08253 1/20 0.49
MMP8 P22894 1/20 0.49
MAPT P10636 2/20 0.48
ALDH1A1 P00352 1/20 0.48
HSD11B1 P28845 1/20 0.46
TRPV1 Q8NER1 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SRD5A2 P31213 1/20 0.46
NR4A1 P22736 1/20 0.45
NR4A2 P43354 1/20 0.45
NR4A3 Q92570 1/20 0.45
PDPK1 O15530 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11137241 0.95 PTPN1 (0.57) PTPN1GSK3BMMP1CES2CES1
SCHEMBL478183 0.85 PTPN1 (0.66) PTPN1GSK3BMMP1CES2CES1
SCHEMBL29987081 0.85 PTPN1 (0.75) PTPN1GSK3BMMP1CES2CES1
SCHEMBL9483307 0.84 MAPT (0.48) PTPN1GSK3BCES1MAPTALDH1A1
SCHEMBL11138890 0.82 PTPN1 (0.54) PTPN1GSK3BMMP1CES2CES1
SCHEMBL3569892 0.81 PTPN1 (0.66) PTPN1GSK3BMMP1CES2CES1
SCHEMBL2269889 0.80 MAPT (0.61) PTPN1GSK3BMMP1CES2CES1
SCHEMBL11132480 0.80 PTPN1 (0.51) PTPN1GSK3BMMP1CES2CES1
SCHEMBL1643579 0.79 PTPN1 (0.73) PTPN1GSK3BMMP1CES2CES1
SCHEMBL6604902 0.79 HTR7 (0.56) PTPN1CES2CES1HDAC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102757-B1 SUBSTITUTED OXAZOLE AND THIAZOLE DERIVATIVES AS HPPAR GAMMA AND HPPAR ALPHA ACTIVATORS GLAXO GROUP LTD (GB) 2004-04-14 EP disclosed